El código ATC L02 La terapia endocrina es un subgrupo terapéutico del Sistema de clasificación química terapéutica anatómica , un sistema de códigos alfanuméricos desarrollado por la Organización Mundial de la Salud (OMS) para la clasificación de medicamentos y otros productos médicos. [1] [2] El subgrupo L02 es parte del grupo anatómico L Antineoplásicos e inmunomoduladores . [3]
Los códigos para uso veterinario ( códigos ATCvet ) se pueden crear colocando la letra Q delante del código ATC humano: por ejemplo, QL02 . [4]
Las cuestiones nacionales de la clasificación ATC pueden incluir códigos adicionales que no están presentes en esta lista, que sigue a la versión de la OMS.
Hormonas L02A y agentes relacionados L02AA01 dietilestilbestrol L02AA02 Fosfato de poliestradiol L02AA03 Etinilestradiol L02AA04 Fosfestrol L02AB01 megestrol L02AB02 medroxiprogesterona L02AB03 Gestonorone L02AE01 Buserelina L02AE02 leuprorelina L02AE03 goserelina L02AE04 triptorelina L02AE05 Histrelina L02AE51 Leuprorelina y bicalutamida L02AX Otras hormonas Antagonistas hormonales L02B y agentes relacionados Antiestrógenos L02BA L02BA01 Tamoxifeno L02BA02 toremifeno L02BA03 Fulvestrant L02BB Antiandrógenos L02BB01 flutamida L02BB02 Nilutamida L02BB03 bicalutamida L02BB04 Enzalutamida L02BB05 Apalutamida L02BB06 Darolutamida Inhibidores de la aromatasa L02BG L02BG01 Aminogluthetimida L02BG02 formestano L02BG03 Anastrozol L02BG04 Letrozol L02BG05 Vorozol L02BG06 Exemestano L02BX Otros antagonistas hormonales y agentes relacionados L02BX01 Abarelix L02BX02 Degarelix L02BX03 Abiraterona Referencias ^ "ATC (sistema de clasificación química terapéutica anatómica) - sinopsis" . Institutos Nacionales de Salud . Consultado el 1 de febrero de 2020 . ^ "ATC-Klassifikation mit definierten Tagesdosen DDD" (en alemán). Instituto Alemán de Documentación e Información Médica . Consultado el 1 de febrero de 2020 . ^ "Índice ATC / DDD 2021: código L02" . Centro Colaborador de la OMS para la Metodología de Estadísticas de Medicamentos. ^ "Índice ATCvet 2021: código QL02" . Centro Colaborador de la OMS para la Metodología de Estadísticas de Medicamentos.
Derivados de testosterona: dipropionato de androstenediolUndecilenato de boldenona Clostebol Acetato de clostebol Caproato de clostebol Propionato de clostebol Acetato de cloxotestosterona Prasterona (dehidroepiandrosterona, DHEA) Prasterone enanthate (DHEA enanthate) Prasterone sulfate (DHEA sulfate) Quinbolone Testosterone# Testosterone esters (e.g., testosterone cypionate, testosterone enanthate, testosterone propionate, testosterone undecanoate, testosterone ester mixtures (Deposterona, Omnadren, Sustanon, Testoviron Depot)) Dihydrotestosterone derivatives: Androstanolone (stanolone, dihydrotestosterone, DHT)Androstanolone esters Bolazine capronate Drostanolone propionate (dromostanolone propionate) Epitiostanol Mepitiostane Mesterolone Metenolone acetate (methenolone acetate) Metenolone enanthate (methenolone enanthate) Stenbolone acetate 19-Nortestosterone derivatives: Bolandiol dipropionateNandrolone esters (e.g., nandrolone decanoate, nandrolone phenylpropionate) Norclostebol Norclostebol acetate Oxabolone cipionate (oxabolone cypionate) Trenbolone acetate Trenbolone hexahydrobenzylcarbonate (trenbolone cyclohexylmethylcarbonate) 17α-Alkylated testosterone derivatives: BolasteroneCalusterone Chlorodehydromethyltestosterone (CDMT) Fluoxymesterone Formebolone Metandienone (methandienone, methandrostenolone) Methandriol (methylandrostenediol) Methandriol bisenanthoyl acetate Methandriol dipropionate Methandriol propionate Methyltestosterone Methyltestosterone 3-hexyl ether Oxymesterone Penmesterol Tiomesterone (thiomesterone) 17α-Alkylated dihydrotestosterone derivatives: AndroisoxazoleFurazabol Mebolazine (dimethazine) Mestanolone Oxandrolone Oxymetholone Stanozolol 17α-Alkylated 19-nortestosterone derivatives: EthylestrenolMibolerone Norethandrolone Normethandrone (methylestrenolone, normethisterone) Propetandrol (propethandrol) 17α-Vinyltestosterone derivatives: Norvinisterone (vinylnortestosterone)17α-Ethynyltestosterone derivatives: DanazolGestrinone Progestins (e.g., ethisterone (ethynyltestosterone), levonorgestrel, norgestrel, norethisterone (norethindrone), lynestrenol, norgestrienone) Tibolone Progesterone derivatives: Medroxyprogesterone acetateAntiestrogens (e.g., tamoxifen, clomifene) GnRH agonists (e.g., GnRH (gonadorelin), leuprorelin) Gonadotropins (e.g., LH, hCG)
Steroidal: Abiraterone acetateCanrenone Chlormadinone acetate Cyproterone acetate Delmadinone acetate Dienogest Drospirenone Medrogestone Megestrol acetate Nomegestrol acetate Osaterone acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: ApalutamideBicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil)
Alfatradiol Dutasteride Epristeride Finasteride Saw palmetto extract Abiraterone acetate Aminoglutethimide Bifluranol Cyproterone acetate Flutamide Ketoconazole Nilutamide Seviteronel† Spironolactone
D2 receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride) Estrogens (e.g., bifluranol, diethylstilbestrol, estradiol, estradiol esters, ethinylestradiol, ethinylestradiol sulfonate, paroxypropione) GnRH agonists (e.g., leuprorelin) GnRH antagonists (e.g., cetrorelix) Progestogens (incl., chlormadinone acetate, cyproterone acetate, hydroxyprogesterone caproate, gestonorone caproate, medroxyprogesterone acetate, megestrol acetate) Androstenedione immunogens: Androvax (androstenedione albumin)Ovandrotone albumin (Fecundin)
# WHO-EM‡ Withdrawn from marketClinical trials:† Phase III§ Never to phase III See also Androgen receptor modulators Estrogens and antiestrogens Progestogens and antiprogestogens List of androgens/anabolic steroids
Steroidal: AlfatradiolCertain androgens/anabolic steroids (e.g., testosterone, testosterone esters, methyltestosterone, metandienone, nandrolone esters) (via estrogenic metabolites) Certain progestins (e.g., norethisterone, noretynodrel, etynodiol diacetate, tibolone) Clomestrone Cloxestradiol acetate Conjugated estriol Conjugated estrogens Epiestriol Epimestrol Esterified estrogens Estetrol† Estradiol Estradiol esters (e.g., estradiol acetate, estradiol benzoate, estradiol cypionate, estradiol enanthate, estradiol undecylate, estradiol valerate, polyestradiol phosphate, estradiol ester mixtures (Climacteron)) Estramustine phosphate Estriol Estriol esters (e.g., estriol succinate, polyestriol phosphate) Estrogenic substances Estrone Estrone estersEstrone sulfate Estropipate (piperazine estrone sulfate) Ethinylestradiol# Ethinylestradiol sulfonate Hydroxyestrone diacetate Mestranol Methylestradiol Moxestrol Nilestriol Prasterone (dehydroepiandrosterone; DHEA)Prasterone enanthate Prasterone sulfate Promestriene Quinestradol Quinestrol Nonsteroidal: BenzestrolBifluranol Chlorotrianisene Dienestrol Diethylstilbestrol (stilbestrol) Diethylstilbestrol esters/ethersDimestrol (diethylstilbestrol dimethyl ether) Fosfestrol (diethylstilbestrol diphosphate) Mestilbol (diethylstilbestrol monomethyl ether) Doisynoestrol (fenocycline) Hexestrol Methallenestril Methestrol (promethestrol)Methestrol dipropionate (promethestrol dipropionate) Paroxypropione Quadrosilan Triphenylbromoethylene Triphenylchloroethylene Zeranol Antiandrogens (e.g., bicalutamide) GnRH agonists (e.g., GnRH (gonadorelin), leuprorelin) Gonadotropins (e.g., FSH, LH)
Acolbifene† Anordrin Bazedoxifene Broparestrol Clomifene# Cyclofenil Enclomifene† Epitiostanol Lasofoxifene Mepitiostane Ormeloxifene Ospemifene Raloxifene Tamoxifen# Toremifene Exclusively antagonistic: FulvestrantNoncompetitive inhibitors: TrilostaneFirst-generation: AminoglutethimideTestolactone Second-generation: FadrozoleFormestane Third-generation: AnastrozoleExemestane Letrozole Androgens/anabolic steroids (e.g., testosterone, testosterone esters, nandrolone esters, oxandrolone, fluoxymesterone) D2 receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride) GnRH agonists (e.g., leuprorelin, goserelin) GnRH antagonists (e.g., cetrorelix, elagolix) Progestogens (e.g., chlormadinone acetate, cyproterone acetate, gestonorone caproate, hydroxyprogesterone caproate, medroxyprogesterone acetate, megestrol acetate) Mixed mechanism of action: DanazolGestrinone Androstenedione immunogens: Androvax (androstenedione albumin)Ovandrotone albumin (Fecundin)
# WHO-EM‡ Withdrawn from marketClinical trials:† Phase III§ Never to phase III See also Estrogen receptor modulators Androgens and antiandrogens Progestogens and antiprogestogens List of estrogens
Progesterone derivatives: ProgesteroneQuingestrone Retroprogesterone derivatives: DydrogesteroneTrengestone 17α-Hydroxyprogesterone (and closely related) derivatives: 17α-Hydroxylated: Acetomepregenol (mepregenol diacetate)Algestone acetophenide (dihydroxyprogesterone acetophenide) Anagestone acetate Chlormadinone acetate Chlormethenmadinone acetate Cyproterone acetate Delmadinone acetate Flugestone acetate (flurogestone acetate) Flumedroxone acetate Hydroxyprogesterone acetate Hydroxyprogesterone caproate Hydroxyprogesterone heptanoate Medroxyprogesterone acetate# Megestrol acetate Melengestrol acetate Methenmadinone acetate Osaterone acetate Pentagestrone acetate Proligestone; 17α-Methylated: Medrogestone; Others: Haloprogesterone 19-Norprogesterone derivatives: 17α-Hydroxylated: Gestonorone caproate (gestronol hexanoate)Nomegestrol acetate Norgestomet Segesterone acetate (nestorone, elcometrine); 17α-Methylated: Demegestone Promegestone Trimegestone Testosterone derivatives: Estranes: DanazolDimethisterone Ethisterone 19-Nortestosterone derivatives: Estranes: AllylestrenolAltrenogest Dienogest Etynodiol diacetate Lynestrenol Norethisterone (norethindrone)# Norethisterone acetate Norethisterone enanthate Noretynodrel Norgesterone Norgestrienone Normethandrone (methylestrenolone) Norvinisterone Oxendolone Quingestanol acetate Tibolone; Gonanes: Desogestrel Etonogestrel Gestodene Gestrinone Levonorgestrel# Norelgestromin Norgestimate Norgestrel Spirolactone derivatives: DrospirenoneOthers: Anabolic–androgenic steroids (e.g., nandrolone and esters, trenbolone and esters, ethylestrenol, norethandrolone, others)
Telapristone§ Ulipristal acetate
# WHO-EM‡ Withdrawn from marketClinical trials:† Phase III§ Never to phase III See also Progesterone receptor modulators Androgens and antiandrogens Estrogens and antiestrogens List of progestogens
Peptide: Azagly-nafarelinBuserelin Deslorelin Fertirelin Gonadorelin Goserelin Histrelin Lecirelin Leuprorelin (leuprolide) Nafarelin Peforelin Triptorelin Peptide: AbarelixCetrorelix Degarelix Ganirelix Non-peptide: ElagolixLinzagolix† Relugolix (+estradiol/norethisterone acetate)
Follicle-stimulating hormone Human chorionic gonadotropin Luteinizing hormone Menotropin Urofollitropin
Sex steroid antagonists (via disinhibition of the HPG axis): Antiandrogens (e.g., flutamide, bicalutamide, enzalutamide)Antiestrogens/SERMs (e.g., tamoxifen, clomifene, enclomifene) Aromatase inhibitors (e.g., anastrozole) GnRH agonists (e.g., GnRH) Sex steroid agonists (via negative feedback on the HPG axis): Androgens/anabolic steroids (e.g., testosterone, nandrolone esters, oxandrolone)D2 receptor antagonists (prolactin releasers) (incl., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride) Estrogens (incl., bifluranol, estradiol, estradiol esters, ethinylestradiol, diethylstilbestrol, paroxypropione) Progestogens (incl. progestins, e.g., chlormadinone acetate, cyproterone acetate, hydroxyprogesterone caproate, gestonorone caproate, medroxyprogesterone acetate, megestrol acetate) Others (mixed or unknown mechanism of action): DanazolGestrinone Metallibure
# WHO-EM‡ Withdrawn from marketClinical trials:† Phase III§ Never to phase III See also GnRH and gonadotropin receptor modulatorsAndrogens and antiandrogens Estrogens and antiestrogens Progestogens and antiprogestogens